Search results for " Oxygen heterocycle"

showing 2 items of 2 documents

A joint experimental and ab initio study on the reactivity of several hydroxy selenides. Stereoselective synthesis of cis-disubstituted tetrahydrofur…

2001

Abstract The reactivity of several hydroxy selenides bearing an ethereal chain with catalytic amounts of perchloric acid in dichloromethane was investigated. Results showed that the position of the oxygen atom with respect to the seleniranium ring was crucial in order to get a good yield of the cyclized product. The factors on which yields of the 5- endo cyclization of the seleniranium ions depend were analysed by ab initio (HF/3-21G ∗ ) studies. An explanation of the different coordinating ability, towards the positively charged selenium atom, of the allylic OMe and homoallylic OH-2 groups was given.

Allylic rearrangementStereochemistryOrganic ChemistryAb initioBiochemistryMedicinal chemistryCatalysischemistry.chemical_compoundchemistrycyclizations oxygen heterocycles selenium theoretical studiesYield (chemistry)Drug DiscoveryReactivity (chemistry)StereoselectivityPerchloric acidDichloromethane
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Synthesis of toxyloxanthone B

2014

A synthesis of the naturally occurring xanthone toxyloxanthone B is described, in which the key step is the regioselective addition of a methyl salicylate to a substituted benzyne, followed by cyclization of the intermediate aryl anion to form the xanthone, the regiochemistry of the aryne addition being confirmed by X-ray crystallography. Subsequent introduction of the pyran ring by [3,3]-rearrangement and deprotection completed the synthesis.

Natural products Xanthones Oxygen heterocycle Benzyne addition Claisen rearrangement.StereochemistryArylOrganic ChemistryRegioselectivitySettore CHIM/06 - Chimica OrganicaRing (chemistry)BiochemistryAryneClaisen rearrangementchemistry.chemical_compoundchemistryPyranDrug DiscoveryXanthone
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